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Azilsartan Medoxomil
  • Synonyms: TAK-491; prodrug of Azilsartan
  • ATC: C09CA09
  • Use: Lorem 
  • Chemical name: Lorem ipsum dolor sit amet, consetetur sadipscing elitr, sed diam
  • Formula: Lorem ipsum dolor sit amet,
  • MW:568.5 g/mol
  • CAS-RN:863031-21-4
  • InChI Key:QJFSABGVXDWMIW-UHFFFAOYSA-N
  • InChI:InChI=1S/C30H24N4O8/c1-​3-​38-​28-​31-​23-​10-​6-​9-​22(27(35)​39-​16-​24-​17(2)​40-​30(37)​41-​24)​25(23)​34(28)​15-​18-​11-​13-​19(14-​12-​18)​20-​7-​4-​5-​8-​21(20)​26-​32-​29(36)​42-​33-​26/h4-​14H,​3,​15-​16H2,​1-​2H3,​(H,​32,​33,​36)

Derivatives

    Azilsartan

  • Use:
  • Formula: Lorem ipsum dolor sit amet,
  • MW:456.5 g/mol
  • CAS-RN:147403-03-0

Substance Classes

Synthesis Path



Substances Referenced in Synthesis Path

CAS-RN Formula Chemical Name CAS Index Name
603-11-2 C8H5NO6 3-nitrophthalic acid
16533-45-2 C10H9NO6 ethyl 2-carboxy-3-nitrobenzoate 1,2-Benzenedicarboxylic acid, 3-nitro-, 1-ethyl ester
136285-65-9 C14H18N2O6 ethyl 2-[(tert-butoxycarbonyl)amino]-3-nitrobenzoate Benzoic acid, 2-[[(1,1-dimethylethoxy)carbonyl]amino]-3-nitro-, ethyl ester
114772-54-2 C14H10BrN 4-(2-cyanobiphenyl)-methyl bromide [1,1'-Biphenyl]-2-carbonitrile, 4'-(bromomethyl)-
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem

Trade Names

Country Trade Name Vendor Annotation
EU Lorem Lorem
USA Lorem Lorem
Lorem Lorem
(wfm = withdrawn from market)

Formulations

  • Loremipsumdolorsitamet,consetetursadipscingelitr,seddiamnonumyeirmodtemporinviduntutlaboreet

References

    • a US 9 999 999 (Takeda; 10.12.1996; appl. 16.8.1994; JP-prior. 25.6.1992).
    • US 9 999 999 (Takeda; 25.8.2005; appl. 7.1.2005; JP-prior. 25.2.2004).
    • US 9 999 999 (Takeda; 14.12.2005; appl. 23.8.2006; JP.-prior. 25.2.2004).
    • b Radl, S. et al., Org. Process Res. Dev., (2013) 17, 77-86.

  • combination with Hydrochlorothiazide:

    • US 9 999 999 (Takeda; 28.9.1999; appl. 26.6.1997; JP-prior. 7.6.1993).

  • alternative synthesis:

    • WO 9999 999999 (Jubilant; 16.8.2012; appl. 24.1.2012; IN-prior. 8.2.2011).
    • WO 9999 999999 (Ranbaxy; 28.3.2012; appl. 20.9.2012; IN-prior. 20.9.2011).

  • solid state forms:

    • WO 9999 999999 (Jubilant; 20.6.2013; appl. 13.12.2012; IN-prior. 15.12.2012).
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