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Tandospirone
  • Synonyms: SM-3997 (as citrate)
  • ATC: N05BX
  • Use: Lorem  Lorem 
  • Chemical name: Lorem ipsum dolor sit amet, consetetur sadipscing elitr, sed diam
  • Formula: Lorem ipsum dolor sit amet,
  • MW:383.50 g/mol
  • CAS-RN:87760-53-0
  • InChI Key:CEIJFEGBUDEYSX-FZDBZEDMSA-N
  • InChI:InChI=1S/C21H29N5O2/c27-​19-​17-​15-​4-​5-​16(14-​15)​18(17)​20(28)​26(19)​9-​2-​1-​8-​24-​10-​12-​25(13-​11-​24)​21-​22-​6-​3-​7-​23-​21/h3,​6-​7,​15-​18H,​1-​2,​4-​5,​8-​14H2/t15-,​16+,​17+,​18-

Derivatives

    citrate

  • Use:
  • Formula: Lorem ipsum dolor sit amet,
  • MW:575.62 g/mol
  • CAS-RN:112457-95-1

Substance Classes

Synthesis Path




Substances Referenced in Synthesis Path

CAS-RN Formula Chemical Name CAS Index Name
628-20-6 C4H6ClN 4-chlorobutyronitrile Butanenitrile, 4-chloro-
14166-28-0 C9H10O3 norbornane-2exo,3exo-dicarboxylic acid anhydride 4,7-Methanoisobenzofuran-1,3-dione, hexahydro-,(3aα,4β,7β,7aα)-
2746-19-2 C9H8O3 norborn-5-ene-2exo,3exo-dicarboxylic acid anhydride 4,7-Methanoisobenzofuran-1,3-dione, 3a,4,7,7a-tetrahydro-,(3aα,4β,7β,7aα)-
20980-22-7 C8H12N4 1-(pyrimidin-2-yl)piperazine Pyrimidine, 2-(1-piperazinyl)-
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem
Lorem Lorem Lorem Lorem

Trade Names

Country Trade Name Vendor Annotation
J Lorem Lorem
(wfm = withdrawn from market)

Formulations

  • Loremipsumdolorsitamet,

References

    • EP 99 999 (Sumitomo Chem.; appl. 29.6.1983; J-prior. 22.12.1981, 3.6.1982).
    • JP 99 999 999 (Sumitomo Chem.; appl. 16.5.1985; USA-prior. 19.1.1983).
    • JP 99 999 999 (Sumitomo Chem.; appl. 18.1.1988; J-prior. 1.7.1986).

  • use of tandospirone: a) treating depression:

    • US 9 999 999 (Pfizer; appl. 30.4.1991; USA-prior. 14.11.1989).

  • b) as psychotropic agents:

    • US 9 999 999 (Bristol-Myers Squibb; appl. 28.5.1996; USA-prior. 5.5.1994).

  • c) as 5-HT1A-receptor agonist:

    • WO 9 999 999 (Medinova SF; appl. 29.2.1996; GB-prior. 23.8.1994).

  • dosage forms:

    • US 9 999 999 (Alza Corp.; appl. 19.7.1994; USA-prior. 27.1.1993).
    • US 9 999 999 (Alza Corp.; appl. 21.9.1993; USA-prior. 27.2.1992, 10.9.1992).
    • US 9 999 999 (Alza Corp.; appl. 22.9.1993; USA-prior. 27.2.1992, 10.9.1992).
    • US 9 999 999 (Alza Corp.; appl. 9.2.1993; USA-prior. 27.2.1992).

  • synergistic compositions with 8-hydroxy-2-(dipropylamino)tetraline and idazoxan:

    • US 9 999 999 (Pfizer; appl. 23.6.1992; USA-prior. 23.4.1991).

  • synthesis of I:

    • Kikuo, I. et al.: Chem. Pharm. Bull. (CPBTAL) 39, 9999 (1991).
    • Wu et al.: J. Med. Chem. (JMCMAR) 15, 999 (1972).
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